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Publication Details
AFRICAN RESEARCH NEXUS
SHINING A SPOTLIGHT ON AFRICAN RESEARCH
medicine
In vitro activity of proveblue (methylene blue) on Plasmodium falciparum strains resistant to standard antimalarial drugs
Antimicrobial Agents and Chemotherapy, Volume 55, No. 5, Year 2011
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Description
The geometric mean 50% inhibitory concentration (IC50) for Proveblue, a methylene blue complying with the European Pharmacopoeia, was more active on 23 P. falciparum strains than chloroquine, quinine, mefloquine, monodesethylamodiaquine, and lumefantrine. We did not find significant associations between the Proveblue IC50 and polymorphisms in the pfcrt, pfmdr1, pfmdr2, pfmrp, and pfnhe-1 genes or the copy numbers of the pfmdr1 and pfmdr2 genes, all of which are involved in antimalarial resistance. Copyright © 2011, American Society for Microbiology. All Rights Reserved.
Authors & Co-Authors
Pascual, Aurélie M.
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Henry, Maud
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Briolant, Sébastien
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Baret, Eric
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Amalvict, Rémy
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Rogier, Christophe
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Pradines, Bruno
France, Marseille
Imtssa Institut de Médecine Tropicale du Service de Santé Des Armées
Statistics
Citations: 55
Authors: 7
Affiliations: 1
Identifiers
Doi:
10.1128/AAC.01466-10
ISSN:
00664804