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Publication Details
AFRICAN RESEARCH NEXUS
SHINING A SPOTLIGHT ON AFRICAN RESEARCH
pharmacology, toxicology and pharmaceutics
Diclofenac sodium delivery to the eye: In vitro evaluation of novel solid lipid nanoparticle formulation using human cornea construct
International Journal of Pharmaceutics, Volume 355, No. 1-2, Year 2008
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Description
Solid lipid nanoparticles (SLNs) were prepared with a combination of homolipid from goat (goat fat) and phospholipid, and evaluated for diclofenac sodium (DNa) delivery to the eye using bio-engineered human cornea, produced from immortalized human corneal endothelial cells (HENC), stromal fibroblasts and epithelial cells CEPI 17 CL 4. Encapsulation efficiency was high and sustained release of DNa and high permeation through the bio-engineered cornea were achieved. Results obtained in this work showed that permeation of DNa through the cornea construct was improved by formulation as SLN modified with phospholipid. © 2007 Elsevier B.V. All rights reserved.
Authors & Co-Authors
Attama Anthony, A. Amaechi
Germany, Braunschweig
Technische Universität Braunschweig
Nigeria, Naukka
University of Nigeria
Reichl, Stephan
Germany, Braunschweig
Technische Universität Braunschweig
Müller-Goymann, Christel Charlotte
Germany, Braunschweig
Technische Universität Braunschweig
Statistics
Citations: 187
Authors: 3
Affiliations: 2
Identifiers
Doi:
10.1016/j.ijpharm.2007.12.007
ISSN:
03785173
Research Areas
Genetics And Genomics
Health System And Policy